Cargando…

Functionalization of α-hydroxyphosphonates as a convenient route to N-tosyl-α-aminophosphonates

Direct conversion of the α-hydroxyl group by para-toluenesulfonamide to yield α-(N-tosyl)aminophosphonates is reported. α-Aminophosphonates 23a,b–37a,b were obtained from the corresponding α-hydroxyphosphonates 6a,b–21a,b in the presence of K(2)CO(3), via the retro-Abramov reaction of the appropriat...

Descripción completa

Detalles Bibliográficos
Autores principales:	Cytlak, Tomasz, Skibińska, Monika, Kaczmarek, Patrycja, Kaźmierczak, Marcin, Rapp, Magdalena, Kubicki, Maciej, Koroniak, Henryk
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	The Royal Society of Chemistry 2018
Materias:	Chemistry
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9079259/ https://www.ncbi.nlm.nih.gov/pubmed/35539392 http://dx.doi.org/10.1039/c8ra01656a

Ejemplares similares

Pyrrolidine and oxazolidine ring transformations in proline and serine derivatives of α-hydroxyphosphonates induced by deoxyfluorinating reagents
por: Kaczmarek, Patrycja, et al.
Publicado: (2018)

Efficient synthesis of dipeptide analogues of α-fluorinated β-aminophosphonates
por: Kaźmierczak, Marcin, et al.
Publicado: (2020)

Highly Diastereoselective Construction of Carbon– Heteroatom Quaternary Stereogenic Centers in the Synthesis of Analogs of Bioactive Compounds: From Monofluorinated Epoxyalkylphosphonates to α-Fluoro-, β-, or γ-Amino Alcohol Derivatives of Alkylphosphonates
por: Rapp, Magdalena, et al.
Publicado: (2021)

Direct Access to Substituted 4-CF(3) β-Lactams at the C-3 Position
por: Skibińska, Monika, et al.
Publicado: (2019)

Synthesis and Reactions of α-Hydroxyphosphonates
por: Rádai, Zita, et al.
Publicado: (2018)

Green and Effective Preparation of α-Hydroxyphosphonates by Ecocatalysis
por: Cybulska, Pola, et al.
Publicado: (2022)

The Stereochemical Course of the α-Hydroxyphosphonate–Phosphate Rearrangement
por: Pallitsch, Katharina, et al.
Publicado: (2015)

Resolution of Racemic α-Hydroxyphosphonates: Bi(OTf)(3)-Catalyzed Stereoselective Esterification of α-Hydroxyphosphonates with (+)-Dibenzoyl-l-tartaric Anhydride
por: Kaboudin, Babak, et al.
Publicado: (2019)

A Highly Efficient Bismuth Salts-Catalyzed Route for the Synthesis of α-Aminophosphonates
por: Banik, Antara, et al.
Publicado: (2010)

Enantioselective dearomatization of isoquinolines by anion-binding catalysis en route to cyclic α-aminophosphonates
por: Ray Choudhury, Abhijnan, et al.
Publicado: (2016)

Novel α-Aminophosphonates and α-Aminophosphonic Acids: Synthesis, Molecular Docking and Evaluation of Antifungal Activity against Scedosporium Species
por: Cordero-Díaz, Anthonny, et al.
Publicado: (2022)

The Last Decade of Optically Active α-Aminophosphonates
por: Varga, Petra R., et al.
Publicado: (2023)

Design, Synthesis, and Antifungal Activity of New α-Aminophosphonates
por: Rezaei, Zahra, et al.
Publicado: (2011)

Asymmetric Synthesis of Tetrasubstituted α-Aminophosphonic Acid Derivatives
por: Maestro, Aitor, et al.
Publicado: (2021)

The synthesis of α-aryl-α-aminophosphonates and α-aryl-α-aminophosphine oxides by the microwave-assisted Pudovik reaction
por: Bálint, Erika, et al.
Publicado: (2017)

Ugi Reaction on α-Phosphorated Ketimines for the Synthesis of Tetrasubstituted α-Aminophosphonates and Their Applications as Antiproliferative Agents
por: López-Francés, Adrián, et al.
Publicado: (2021)

α-Aminophosphonate Derivatives for Enhanced Flame Retardant Properties in Epoxy Resin
por: Stanfield, Melissa K., et al.
Publicado: (2021)

Synthesis of Novel 1,3,4-Oxadiazole-Derived α-Aminophosphonates/α-Aminophosphonic Acids and Evaluation of Their In Vitro Antiviral Activity against the Avian Coronavirus Infectious Bronchitis Virus
por: Hkiri, Shaima, et al.
Publicado: (2022)

Dipeptide analogues of fluorinated aminophosphonic acid sodium salts as moderate competitive inhibitors of cathepsin C
por: Wątroba, Karolina, et al.
Publicado: (2023)

Synthesis of α-Aminophosphonates and Related Derivatives; The Last Decade of the Kabachnik–Fields Reaction
por: Varga, Petra R., et al.
Publicado: (2021)

One-pot synthesis of α-aminophosphonates by yttrium-catalyzed Birum–Oleksyszyn reaction
por: Ceradini, Davide, et al.
Publicado: (2021)

α-Aminophosphonate inhibitors of metallo-β-lactamases NDM-1 and VIM-2
por: Palica, Katarzyna, et al.
Publicado: (2023)

Transdermal Delivery of α-Aminophosphonates as Semisolid Formulations—An In Vitro-Ex Vivo Study
por: Kocsis, Dorottya, et al.
Publicado: (2023)

Comparative Studies on Regioselectivity of α- and β-Linked Glucan Tosylation
por: Koschella, Andreas, et al.
Publicado: (2020)

A convenient route to optically pure α-alkyl-β-(sec-amino)alanines
por: Olma, A., et al.
Publicado: (2011)

Effect of Microgravity on Fungistatic Activity of an α-Aminophosphonate Chitosan Derivative against Aspergillus niger
por: Devarayan, Kesavan, et al.
Publicado: (2015)

Synthesis of (R)- and (S)-β-hydroxyphosphonate acyclonucleosides: structural analogues of Adefovir (PMEA)
por: Kasthuri, Mahesh, et al.
Publicado: (2011)

Catalyst-Free Cross-Dehydrogenative Coupling Strategy Using Air as an Oxidant: Synthesis of α-Aminophosphonates
por: Dhineshkumar, Jayaraman, et al.
Publicado: (2017)

Asymmetric Synthesis of α-Aminophosphonates Using the Inexpensive Chiral Catalyst 1,1’-Binaphthol Phosphate
por: Xu, Weiming, et al.
Publicado: (2010)

Cytotoxic Activity of α-Aminophosphonic Derivatives Coming from the Tandem Kabachnik–Fields Reaction and Acylation
por: Varga, Petra R., et al.
Publicado: (2023)

β-Carboline-α-aminophosphonate Derivative: A Promising Antitumor Agent for Breast Cancer Treatment
por: Zani, Caroline Pinto, et al.
Publicado: (2023)

Aromatic fluorocopolymers based on α-(difluoromethyl)styrene and styrene: synthesis, characterization, and thermal and surface properties
por: Wolska, Joanna, et al.
Publicado: (2018)

Silver(I) Complexes Based on Oxadiazole-Functionalized α-Aminophosphonate: Synthesis, Structural Study, and Biological Activities
por: Hkiri, Shaima, et al.
Publicado: (2022)

Synthesis and Characterization of a New Series of Bis(allylic-α-aminophosphonates) under Mild Reaction Conditions
por: Souii, Ichrak, et al.
Publicado: (2023)

Evaluation of Antibacterial Activity against Nosocomial Pathogens of an Enzymatically Derived α-Aminophosphonates Possessing Coumarin Scaffold
por: Kowalczyk, Paweł, et al.
Publicado: (2023)

Discovery of Novel α-Aminophosphonates with Hydrazone as Potential Antiviral Agents Combined With Active Fragment and Molecular Docking
por: Tian, Jia, et al.
Publicado: (2022)

Naphthalene vs. Benzene as a Transmitting Moiety: Towards the More Sensitive Trifluoromethylated Molecular Probes for the Substituent Effects
por: Sokół, Adam, et al.
Publicado: (2022)

Chelating Tendencies of Bioactive Aminophosphonates
por: Kiss, Tamas, et al.
Publicado: (1994)

(25R)-6α-Hydroxy-5α-spirostan-3β-yl tosylate
por: Fernández-Herrera, María A., et al.
Publicado: (2012)

The Synthesis of α-Aminophosphonates via Enantioselective Organocatalytic Reaction of 1-(N-Acylamino)alkylphosphonium Salts with Dimethyl Phosphite
por: Walęcka-Kurczyk, Alicja, et al.
Publicado: (2020)

Cannot write session to /tmp/vufind_sessions/sess_suc892d4k60vc4mq2sguo86fmk