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Palladium-catalyzed intramolecular C–H arylation of 2-halo-N-Boc-N-arylbenzamides for the synthesis of N–H phenanthridinones

A palladium catalyzed synthesis of N–H phenanthridinones was developed via C–H arylation. The protocol gives phenanthridinones regioselectively by one-pot reaction without deprotection. It exhibits broad substrate scope and affords targets in up to 95% yields. Importantly, it could be applied for th...

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Detalles Bibliográficos
Autores principales: Hu, Quan-Fang, Gao, Tian-Tao, Shi, Yao-Jie, Lei, Qian, Yu, Luo-Ting
Formato: Online Artículo Texto
Lenguaje:English
Publicado: The Royal Society of Chemistry 2018
Materias:
Acceso en línea:https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9079793/
https://www.ncbi.nlm.nih.gov/pubmed/35539333
http://dx.doi.org/10.1039/c8ra02099j