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Perspective on the Relationship between GABA(A) Receptor Activity and the Apparent Potency of an Inhibitor
Background: In electrophysiological experiments, inhibition of a receptor-channel, such as the GABA(A) receptor, is measured by co-applying an agonist producing a predefined control response with an inhibitor to calculate the fraction of the control response remaining in the presence of the inhibito...
Autores principales: | Germann, Allison L., Pierce, Spencer R., Evers, Alex S., Steinbach, Joe Henry, Akk, Gustav |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
Bentham Science Publishers
2022
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9199547/ https://www.ncbi.nlm.nih.gov/pubmed/34784870 http://dx.doi.org/10.2174/1570159X19666211104142433 |
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