Optimization of Peptide Linker-Based Fluorescent Ligands for the Histamine H(1) Receptor

[Image: see text] The histamine H(1) receptor (H(1)R) has recently been implicated in mediating cell proliferation and cancer progression; therefore, high-affinity H(1)R-selective fluorescent ligands are desirable tools for further investigation of this behavior in vitro and in vivo. We previously r...

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Detalles Bibliográficos
Autores principales: Kok, Zhi Yuan, Stoddart, Leigh A., Mistry, Sarah J., Mocking, Tamara A. M., Vischer, Henry F., Leurs, Rob, Hill, Stephen J., Mistry, Shailesh N., Kellam, Barrie
Formato: Online Artículo Texto
Lenguaje:English
Publicado: American Chemical Society 2022
Acceso en línea:https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9234962/
https://www.ncbi.nlm.nih.gov/pubmed/35734860
http://dx.doi.org/10.1021/acs.jmedchem.2c00125

Internet

https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9234962/
https://www.ncbi.nlm.nih.gov/pubmed/35734860
http://dx.doi.org/10.1021/acs.jmedchem.2c00125

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