Cargando…
Chemical Exploration of a Highly Selective Scaffold with Activity against Intracellular Mycobacterium tuberculosis
We previously identified a phenylthiourea series with activity against intracellular Mycobacterium tuberculosis using a high-throughput, high-content assay. We conducted a catalog structure-activity relationship study with a collection of 35 analogs. We identified several thiourea derivatives with e...
Autores principales: | Njikan, Samuel, Ahmed, Sara, Manning, Alyssa, Awasthi, Divya, Ovechkina, Yulia, Chowdhury, Sultan, Butts, Arielle, Parish, Tanya |
---|---|
Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
American Society for Microbiology
2022
|
Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9241686/ https://www.ncbi.nlm.nih.gov/pubmed/35612308 http://dx.doi.org/10.1128/spectrum.01161-22 |
Ejemplares similares
-
Identification of Novel Chemical Scaffolds that Inhibit the Growth of Mycobacterium tuberculosis in Macrophages
por: Ahmed, Sara, et al.
Publicado: (2022) -
High content, high-throughput screening for small molecule inducers of NF-κB translocation
por: Njikan, Samuel, et al.
Publicado: (2018) -
Benzene Amide
Ether Scaffold is Active against Non-replicating
and Intracellular Mycobacterium tuberculosis
por: Ahmed, Sara, et al.
Publicado: (2023) -
Triazolopyrimidines Target Aerobic Respiration in Mycobacterium tuberculosis
por: Shelton, Catherine, et al.
Publicado: (2022) -
Identification of 2-Amino Benzothiazoles with Bactericidal Activity against Mycobacterium tuberculosis
por: Bonnett, Shilah, et al.
Publicado: (2023)