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Screening of Hydrocarbon-Stapled Peptides for Inhibition of Calcium-Triggered Exocytosis
The so-called primary interface between the SNARE complex and synaptotagmin-1 (Syt1) is essential for Ca(2+)-triggered neurotransmitter release in neuronal synapses. The interacting residues of the primary interface are conserved across different species for synaptotagmins (Syt1, Syt2, Syt9), SNAP-2...
Autores principales: | Lai, Ying, Tuvim, Michael J., Leitz, Jeremy, Peters, John, Pfuetzner, Richard A., Esquivies, Luis, Zhou, Qiangjun, Czako, Barbara, Cross, Jason B., Jones, Philip, Dickey, Burton F., Brunger, Axel T. |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
Frontiers Media S.A.
2022
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9258623/ https://www.ncbi.nlm.nih.gov/pubmed/35814209 http://dx.doi.org/10.3389/fphar.2022.891041 |
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