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Structural determinants of TRPV4 inhibition and identification of new antagonists with antiviral activity
BACKGROUND AND PURPOSE: The transient receptor potential vanilloid 4 (TRPV4) cation channel participates in multiple physiological processes and is also at the core of different diseases, making this channel an interesting pharmacological target with therapeutic potential. However, little is known a...
Autores principales: | Doñate‐Macian, Pablo, Duarte, Yorley, Rubio‐Moscardo, Fanny, Pérez‐Vilaró, Gemma, Canan, Jonathan, Díez, Juana, González‐Nilo, Fernando, Valverde, Miguel A. |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
John Wiley and Sons Inc.
2020
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9291951/ https://www.ncbi.nlm.nih.gov/pubmed/32959389 http://dx.doi.org/10.1111/bph.15267 |
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