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Systematic Evaluation of Fluorination as Modification for Peptide‐Based Fusion Inhibitors against HIV‐1 Infection

With the emergence of novel viruses, the development of new antivirals is more urgent than ever. A key step in human immunodeficiency virus type 1 (HIV‐1) infection is six‐helix bundle formation within the envelope protein subunit gp41. Selective disruption of bundle formation by peptides has been s...

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Detalles Bibliográficos
Autores principales:	Huhmann, Susanne, Nyakatura, Elisabeth K., Rohrhofer, Anette, Moschner, Johann, Schmidt, Barbara, Eichler, Jutta, Roth, Christian, Koksch, Beate
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	John Wiley and Sons Inc. 2021
Materias:	Full Papers
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9297971/ https://www.ncbi.nlm.nih.gov/pubmed/34605595 http://dx.doi.org/10.1002/cbic.202100417

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