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Site‐Selective Pd‐Catalyzed C(sp(3))−H Arylation of Heteroaromatic Ketones

A ligand‐controlled site‐selective C(sp(3))−H arylation of heteroaromatic ketones has been developed using Pd catalysis. The reaction occurred selectively at the α‐ or β‐position of the ketone side‐chain. The switch from α‐ to β‐arylation was realized by addition of a pyridone ligand. The α‐arylatio...

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Detalles Bibliográficos
Autores principales:	Kudashev, Anton, Baudoin, Olivier
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	John Wiley and Sons Inc. 2021
Materias:	Full Papers
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9299137/ https://www.ncbi.nlm.nih.gov/pubmed/34761844 http://dx.doi.org/10.1002/chem.202103467

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