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Asymmetrically Substituted m‐Terphenyl Phosphates Inhibit the Transcription Factor STAT5a
We recently presented Stafia‐1 as the first chemical entity that inhibits the transcription factor STAT5a with selectivity over the highly homologous STAT5b. Stafia‐1, which was identified from a series of symmetrically substituted m‐terphenyl phosphates, binds to the interface between the SH2 domai...
Autores principales: | Müller‐Klieser, Daniel, Berg, Thorsten |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
John Wiley and Sons Inc.
2021
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9303812/ https://www.ncbi.nlm.nih.gov/pubmed/34905258 http://dx.doi.org/10.1002/cbic.202100603 |
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