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Hydrochloride Salt of the GABAkine KRM-II-81
[Image: see text] Imidazodiazepine (5-(8-ethynyl-6-(pyridin-2-yl)-4H-benzo[f]imidazole[1,5-α][1,4]diazepin-3-yl) oxazole or KRM-II-81) is a potentiator of GABA(A) receptors (a GABAkine) undergoing preparation for clinical development. KRM-II-81 is active against many seizure and pain models in roden...
Autores principales: | , , , , , , , , , , , , , , , , |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
American Chemical Society
2022
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Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9366947/ https://www.ncbi.nlm.nih.gov/pubmed/35967038 http://dx.doi.org/10.1021/acsomega.2c03029 |