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Design and Validation of the First Family of Photo-Activatable Ligands for Melatonin Receptors

[Image: see text] Melatonin is a neurohormone released in a circadian manner with peak levels at night. Melatonin mediates its effects mainly through G protein-coupled MT(1) and MT(2) receptors. Drugs acting on melatonin receptors are indicated for circadian rhythm- and sleep-related disorders. Tool...

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Detalles Bibliográficos
Autores principales:	Somalo-Barranco, Gloria, Serra, Carme, Lyons, David, Piggins, Hugh D., Jockers, Ralf, Llebaria, Amadeu
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	American Chemical Society 2022
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9421648/ https://www.ncbi.nlm.nih.gov/pubmed/35930058 http://dx.doi.org/10.1021/acs.jmedchem.2c00717

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