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Discovery of novel conjugates of quinoline and thiazolidinone urea as potential anti-colorectal cancer agent

Based on the obtained SARs, further structural optimisation of compound BC2021-104511-15i was conducted in this investigation, and totally ten novel quinoline derivates were designed, synthesised and optimised for biological activity. Among them, compound 10a displayed significant in vitro anticance...

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Detalles Bibliográficos
Autores principales:	Xiong, Li, He, Huan, Fan, Mengmeng, Hu, Liping, Wang, Fei, Song, Xiaomeng, Shi, Shengmin, Qi, Baohui
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	Taylor & Francis 2022
Materias:	Research Paper
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9448386/ https://www.ncbi.nlm.nih.gov/pubmed/36043496 http://dx.doi.org/10.1080/14756366.2022.2117318

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