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Conjugation of a Cationic Cell-Penetrating Peptide with a Novel Kunitzin-like Trypsin Inhibitor: New Insights for Enhancement of Peptide Bioactivities

Cationic cell-penetrating peptides (CPPs), such as transactivator of transcription (TAT) peptide, have been proposed as effective drug carriers to improve intracellular delivery of biological macromolecules. Amphibian skin-derived Kunitz-type trypsin inhibitors (KTIs), short counterparts of KTIs fro...

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Detalles Bibliográficos
Autores principales: Yao, Junting, Yin, Weining, Chen, Yuqing, Chen, Xiaoling, Jiang, Yangyang, Wang, Tao, Ma, Chengbang, Zhou, Mei, Chen, Tianbao, Shaw, Chris, Wang, Lei
Formato: Online Artículo Texto
Lenguaje:English
Publicado: MDPI 2022
Materias:
Acceso en línea:https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9501525/
https://www.ncbi.nlm.nih.gov/pubmed/36145553
http://dx.doi.org/10.3390/pharmaceutics14091805