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Design, Synthesis, and Bioactivities of Novel Tryptophan Derivatives Containing 2,5-Diketopiperazine and Acyl Hydrazine Moieties

Based on the scaffolds widely used in drug design, a series of novel tryptophan derivatives containing 2,5-diketopiperazine and acyl hydrazine moieties have been designed, synthesized, characterized, and evaluated for their biological activities. The bioassay results showed that the target compounds...

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Detalles Bibliográficos
Autores principales:	Li, Lili, Yang, Rongxin, Liu, Jianhua, Zhang, Jingjing, Song, Hongjian, Liu, Yuxiu, Wang, Qingmin
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	MDPI 2022
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9506431/ https://www.ncbi.nlm.nih.gov/pubmed/36144506 http://dx.doi.org/10.3390/molecules27185758

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