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Apamin structure and pharmacology revisited
Apamin is often cited as one of the few substances selectively acting on small-conductance Ca(2+)-activated potassium channels (K(Ca)2). However, published pharmacological and structural data remain controversial. Here, we investigated the molecular pharmacology of apamin by two-electrode voltage-cl...
Autores principales: | Kuzmenkov, Alexey I., Peigneur, Steve, Nasburg, Joshua A., Mineev, Konstantin S., Nikolaev, Maxim V., Pinheiro-Junior, Ernesto Lopes, Arseniev, Alexander S., Wulff, Heike, Tytgat, Jan, Vassilevski, Alexander A. |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
Frontiers Media S.A.
2022
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9523135/ https://www.ncbi.nlm.nih.gov/pubmed/36188602 http://dx.doi.org/10.3389/fphar.2022.977440 |
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