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Guanidine Derivatives of Quinazoline-2,4(1H,3H)-Dione as NHE-1 Inhibitors and Anti-Inflammatory Agents

Quinazolines are a rich source of bioactive compounds. Previously, we showed NHE-1 inhibitory, anti-inflammatory, antiplatelet, intraocular pressure lowering, and antiglycating activity for a series of quinazoline-2,4(1H,3H)-diones and quinazoline-4(3H)-one guanidine derivatives. In the present work...

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Detalles Bibliográficos
Autores principales: Spasov, Alexander, Ozerov, Alexander, Kosolapov, Vadim, Gurova, Natalia, Kucheryavenko, Aida, Naumenko, Ludmila, Babkov, Denis, Sirotenko, Viktor, Taran, Alena, Borisov, Alexander, Sokolova, Elena, Klochkov, Vladlen, Merezhkina, Darya, Miroshnikov, Mikhail, Ovsyankina, Nadezhda, Smirnov, Alexey, Velikorodnaya, Yulia
Formato: Online Artículo Texto
Lenguaje:English
Publicado: MDPI 2022
Materias:
Acceso en línea:https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9605072/
https://www.ncbi.nlm.nih.gov/pubmed/36295082
http://dx.doi.org/10.3390/life12101647