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Design, Synthesis, In Silico Testing, and In Vitro Evaluation of Thiazolidinone-Based Benzothiazole Derivatives as Inhibitors of α-Amylase and α-Glucosidase
In this study, a stepwise reaction afforded thiazolidinone-based benzothiazole derivatives 1–15, and the synthesized derivatives were then screened for biological significance and found to be the leading candidates against α-amylase and α-glucosidase enzymes. Almost all derivatives showed excellent...
Autores principales: | Khan, Shoaib, Iqbal, Shahid, Khan, Marwa, Rehman, Wajid, Shah, Mazloom, Hussain, Rafaqat, Rasheed, Liaqat, Khan, Yousaf, Dera, Ayed A., Pashameah, Rami Adel, Alzahrani, Eman, Farouk, Abd-ElAziem |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
MDPI
2022
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9610606/ https://www.ncbi.nlm.nih.gov/pubmed/36297276 http://dx.doi.org/10.3390/ph15101164 |
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