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Structural basis of organic cation transporter-3 inhibition

Organic cation transporters (OCTs) facilitate the translocation of catecholamines, drugs and xenobiotics across the plasma membrane in various tissues throughout the human body. OCT3 plays a key role in low-affinity, high-capacity uptake of monoamines in most tissues including heart, brain and liver...

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Detalles Bibliográficos
Autores principales: Khanppnavar, Basavraj, Maier, Julian, Herborg, Freja, Gradisch, Ralph, Lazzarin, Erika, Luethi, Dino, Yang, Jae-Won, Qi, Chao, Holy, Marion, Jäntsch, Kathrin, Kudlacek, Oliver, Schicker, Klaus, Werge, Thomas, Gether, Ulrik, Stockner, Thomas, Korkhov, Volodymyr M., Sitte, Harald H.
Formato: Online Artículo Texto
Lenguaje:English
Publicado: Nature Publishing Group UK 2022
Materias:
Acceso en línea:https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9640557/
https://www.ncbi.nlm.nih.gov/pubmed/36344565
http://dx.doi.org/10.1038/s41467-022-34284-8