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Acetylation Enhances the Anticancer Activity and Oral Bioavailability of 5-Demethyltangeretin

A kind of hydroxylated polymethoxyflavone (PMFs) existing in the citrus genus, 5-Demethyltangeretin (5-DTAN), has been reported to possess several bioactivities in vitro and in vivo. The aim of this study was to investigate whether acetylation could enhance the anticancer activity and oral bioavaila...

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Detalles Bibliográficos
Autores principales: Tsai, Hui-Yun, Yang, Jia-Fang, Chen, Yin-Bo, Guo, Jia-Lin, Li, Shiming, Wei, Guor-Jien, Ho, Chi-Tang, Hsu, Jue-Liang, Chang, Chi-I, Liang, Yu-Shen, Yu, Hsu-Sheng, Chen, Yu-Kuo
Formato: Online Artículo Texto
Lenguaje:English
Publicado: MDPI 2022
Materias:
Acceso en línea:https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9658984/
https://www.ncbi.nlm.nih.gov/pubmed/36362072
http://dx.doi.org/10.3390/ijms232113284