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Insights into Antimalarial Activity of N-Phenyl-Substituted Cinnamanilides
Due to the urgent need of innovation in the antimalarial therapeutic arsenal, a series of thirty-seven ring-substituted N-arylcinnamanilides prepared by microwave-assisted synthesis were subjected to primary screening against the chloroquine-sensitive strain of P. falciparum 3D7/MRA-102. The lipophi...
Autores principales: | Kos, Jiri, Degotte, Gilles, Pindjakova, Dominika, Strharsky, Tomas, Jankech, Timotej, Gonec, Tomas, Francotte, Pierre, Frederich, Michel, Jampilek, Josef |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
MDPI
2022
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9698057/ https://www.ncbi.nlm.nih.gov/pubmed/36431900 http://dx.doi.org/10.3390/molecules27227799 |
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