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Estrogen Receptor-α Targeting: PROTACs, SNIPERs, Peptide-PROTACs, Antibody Conjugated PROTACs and SNIPERs

Targeting selective estrogen subtype receptors through typical medicinal chemistry approaches is based on occupancy-driven pharmacology. In occupancy-driven pharmacology, molecules are developed in order to inhibit the protein of interest (POI), and their popularity is based on their virtue of faste...

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Detalles Bibliográficos
Autores principales: Negi, Arvind, Kesari, Kavindra Kumar, Voisin-Chiret, Anne Sophie
Formato: Online Artículo Texto
Lenguaje:English
Publicado: MDPI 2022
Materias:
Acceso en línea:https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9699327/
https://www.ncbi.nlm.nih.gov/pubmed/36432713
http://dx.doi.org/10.3390/pharmaceutics14112523