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Development of Novel Isatin-Tethered Quinolines as Anti-Tubercular Agents against Multi and Extensively Drug-Resistant Mycobacterium tuberculosis

We describe the design and synthesis of two isatin-tethered quinolines series (Q6a–h and Q8a–h), in connection with our research interest in developing novel isatin-bearing anti-tubercular candidates. In a previous study, a series of small molecules bearing a quinoline-3-carbohydrazone moiety was de...

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Detalles Bibliográficos
Autores principales: Abdelrahman, Mohamed A., Almahli, Hadia, Al-Warhi, Tarfah, Majrashi, Taghreed A., Abdel-Aziz, Marwa M., Eldehna, Wagdy M., Said, Mohamed A.
Formato: Online Artículo Texto
Lenguaje:English
Publicado: MDPI 2022
Materias:
Acceso en línea:https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9781264/
https://www.ncbi.nlm.nih.gov/pubmed/36557937
http://dx.doi.org/10.3390/molecules27248807