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Synthesis and Antiprotozoal Activity of Azabicyclo-Nonane Pyrimidine Hybrids

2,4-Diaminopyrimidines and (dialkylamino)azabicyclo-nonanes possess activity against protozoan parasites. A series of fused hybrids were synthesized and tested in vitro against pathogens of malaria tropica and sleeping sickness. The activities and selectivities of compounds strongly depended on the...

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Detalles Bibliográficos
Autores principales:	Hinteregger, Clemens, Dolensky, Johanna, Seebacher, Werner, Saf, Robert, Mäser, Pascal, Kaiser, Marcel, Weis, Robert
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	MDPI 2022
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9821907/ https://www.ncbi.nlm.nih.gov/pubmed/36615504 http://dx.doi.org/10.3390/molecules28010307

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