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Click-designed vanilloid-triazole conjugates as dual inhibitors of AChE and Aβ aggregation
Based on their reported neuroprotective properties, vanilloids provide a good starting point for the synthesis of anti-Alzheimer's disease (AD) agents. In this context, nine new 1,2,3-triazole conjugates of vanilloids were synthesized via click chemistry. The compounds were tested for their eff...
Autores principales: | Elsbaey, Marwa, Igarashi, Yasuhiro, Ibrahim, Mahmoud A. A., Elattar, Eman |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
The Royal Society of Chemistry
2023
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9850456/ https://www.ncbi.nlm.nih.gov/pubmed/36756452 http://dx.doi.org/10.1039/d2ra07539c |
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