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Synthesis and characterisation of new antimalarial fluorinated triazolopyrazine compounds

Nine new fluorinated analogues were synthesised by late-stage functionalisation using Diversinate™ chemistry on the Open Source Malaria (OSM) triazolopyrazine scaffold (Series 4). The structures of all analogues were fully characterised by NMR, UV and MS data analysis; three triazolopyrazines were c...

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Detalles Bibliográficos
Autores principales:	Lum, Kah Yean, White, Jonathan M, Johnson, Daniel J G, Avery, Vicky M, Davis, Rohan A
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	Beilstein-Institut 2023
Materias:	Full Research Paper
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9907012/ https://www.ncbi.nlm.nih.gov/pubmed/36761470 http://dx.doi.org/10.3762/bjoc.19.11

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