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(68)Ga-Labeled [Thz(14)]Bombesin(7–14) Analogs: Promising GRPR-Targeting Agonist PET Tracers with Low Pancreas Uptake

With overexpression in various cancers, the gastrin-releasing peptide receptor (GRPR) is a promising target for cancer imaging and therapy. However, the high pancreas uptake of reported GRPR-targeting radioligands limits their clinical application. Our goal was to develop (68)Ga-labeled agonist trac...

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Detalles Bibliográficos
Autores principales:	Wang, Lei, Bratanovic, Ivica Jerolim, Zhang, Zhengxing, Kuo, Hsiou-Ting, Merkens, Helen, Zeisler, Jutta, Zhang, Chengcheng, Tan, Ruiyan, Bénard, François, Lin, Kuo-Shyan
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	MDPI 2023
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9962964/ https://www.ncbi.nlm.nih.gov/pubmed/36838968 http://dx.doi.org/10.3390/molecules28041977

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