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Structure–Activity Relationship and Evaluation of Phenethylamine and Tryptamine Derivatives for Affinity towards 5-Hydroxytryptamine Type 2A Receptor

Among 14 subtypes of serotonin receptors (5-HTRs), 5-HT(2A)R plays important roles in drug addiction and various psychiatric disorders. Agonists for 5-HT(2A)R have been classified into three structural groups: phenethylamines, tryptamines, and ergolines. In this study, the structure-activity relatio...

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Detalles Bibliográficos
Autores principales:	Wang, Shujie, Zhu, Anlin, Paudel, Suresh, Jang, Choon-Gon, Lee, Yong Sup, Kim, Kyeong-Man
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	The Korean Society of Applied Pharmacology 2023
Materias:	Original Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9970836/ https://www.ncbi.nlm.nih.gov/pubmed/36224112 http://dx.doi.org/10.4062/biomolther.2022.096

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